HyperLab Main Feature Update History

This information pertains to updates in HyperLab that may have affected users’ calculation results.

1. Hyper Binding

Update Date
HyperLab Version
Changelog
Description
Release Note

March 28, 2024

2024.03.28

ES update

  1. Exhaustive Search, our brand-new development of a binding-pose search method, and

  2. PIGNet2, our published AI for predicting protein-ligand interactions [Digital Discovery 3: 287 (2024)].

  3. Exhaustive Search significantly increases both Hyper Binding's accuracy and speed.

October 18, 2024

2024.10.18

Improved Hyper Binding success rate

The calculation success rate of Hyper Binding has been enhanced.

November 15, 2024

2024.11.15

Improved ligand ionization handling

Corrected the ionized forms of some functional groups of ligands.

April 10, 2025

2025.04.10

Update with applied Box size calculation method

For proteins registered as 3D Structure type, the box size you set is now more precisely reflected in calculations.

2. Hyper ADME/T

Update Date
HyperLab Version
Changelog
Description
Release Note

October 18, 2024

2024.10.18

Changes to the Metabolic stability

The Metabolic stability in Hyper ADME/T is now changed to Metabolic stability (H/M).

3. Hyper Design

Update Date
HyperLab Version
Changelog
Description
Release Note

August 30, 2024

2024.08.30

Changing the physicochemical property values of some molecules

The physicochemical property values of ionizable molecules added by hyperdesign have been changed.

October 18, 2024

2024.10.18

Added R group definition feature

In Hyper Design, you can now define the fragment design to a specific R-group. (Examples of R-groups: Aliphatic chains, Aryl, Heteroaryl, etc.)

November 15, 2024

2024.11.15

Performance improvement

  1. The multiple selection bug in the fragment library has been fixed.

  2. The Hyder Design algorithm has been improved to allow ‘Add’ feature to bond with carbons that have double bonds.

4. Hyper Screening

Update Date
HyperLab Version
Changelog
Description
Release Note

August 9, 2024

2024.08.09

PAINS Filter applied

The PAINS (Pan-Assay Interference Compounds) filter has been applied to the HyperLab library.

5. 3D Viewer

Update Date
HyperLab Version
Changelog
Description
Release Note

November 15, 2024

2024.11.15

Interaction improvement

Enhanced to analyze interaction information with DNA/RNA receptors.

6. Hyper Binding Co-folding

Update Date
HyperLab Version
Changelog
Description
Release Note

April 10, 2025

2025.04.10

New Feature Added

The Hyper Binding Co-folding feature has been newly added.

7. Hyper Screening X

Update Date
HyperLab Version
Changelog
Description
Release Note

April 10, 2025

2025.04.10

New Feature Added

The Hyper Screening X feature has been newly added.

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